Kuehne, Martin et al. published their patent in 1990 |CAS: 42900-89-0

The Article related to vinblastine cycloalkyl aryl preparation antitumor, cycloalkylvinblastine preparation antitumor, vincristine cycloalkyl aryl preparation antitumor, cycloalkylvincristine preparation antitumor, antitumor vinblastine vincristine cycloalkyl aryl, arylvinblastine preparation antitumor, arylvincristine preparation antitumor and other aspects.Safety of Isochroman-3-ol

On June 19, 1990, Kuehne, Martin published a patent.Safety of Isochroman-3-ol The title of the patent was Preparation of cycloalkyl and aromatic moieties-containing vinblastines and vincristines as antitumors. And the patent contained the following:

The title compounds [I; R1R2 = alkylene, benzo; R10 = HCO, Me; R11 = alkoxy, trialkylammoniumyl; R12 = alkanoyloxy, OH; R13 = alkyl] were prepared Vindoline-HCl was condensed with Me (3aRS,4RS,11bSR)]-3-benzyl-4-[2-(tert-butyldimethylsilyloxymethyl)phenyl]-1,2,3,3a,4,5-hexahydro-7H-pyrrolo[2,3-d]carbazole-6-carboxylate to give, after desilylation, a 1:1 mixture of (5R,7S)-3-benzyl-5-[2-(hydroxymethyl)phenyl]-1,2,3,4,5,6,7,8-octahydroazonino[5,4-b]indole-7-(15-vindolinyl)-7-carboxylate (II) and its 5R,7R-diastereomer. II was then cyclized in CH2Cl2 containing Et3N and p-toluenesulfonic anhydride to give, after hydrogenolysis, (9R,11S)-15-[1,2,4,9,10,11,12,17-octahydro-11-(methoxycarbonyl)indolo[2′,3′:6,7]azonino[1,2,3:bc]isoquinolin-11-yl]vindoline (III). III had an ED50 comparable to that of vinblastine against P388 leukemia cells resistant to adriamycin. The experimental process involved the reaction of Isochroman-3-ol(cas: 42900-89-0).Safety of Isochroman-3-ol

The Article related to vinblastine cycloalkyl aryl preparation antitumor, cycloalkylvinblastine preparation antitumor, vincristine cycloalkyl aryl preparation antitumor, cycloalkylvincristine preparation antitumor, antitumor vinblastine vincristine cycloalkyl aryl, arylvinblastine preparation antitumor, arylvincristine preparation antitumor and other aspects.Safety of Isochroman-3-ol

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